Description：

CH5132799 inhibits class I PI3Ks, particularly PI3Kα with IC50 of 14 nM; less potent to PI3Kβδγ, while sensitive in PIK3CA mutations cell lines. Phase 1.

Chemical Information：

Molecular Weight (MW)		377.42
Formula		C15H19N7O3S
CAS No.		1007207-67-1
Solubility (25°C) *	DMSO	12 mg/mL (31.79 mM)
	Water	Insoluble
	Alcohol	Insoluble

Biological Activity：

Targets IC50

GPR40 14 nM (EC50) [1

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	2.6496 mL	13.2478 mL	26.4957 mL
5 mM	0.5299 mL	2.6496 mL	5.2991 mL
10 mM	0.2650 mL	1.3248 mL	2.6496 mL
50 mM	0.0530 mL	0.2650 mL	0.5299 mL

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