Description：

BMS-754807 is a potent and reversible inhibitor of IGF-1R/InsR with IC50 of 1.8 nM/1.7 nM in cell-free assays, less potent to Met, Aurora A/B, TrkA/B and Ron, and shows little activity to Flt3, Lck, MK2, PKA, PKC etc. Phase 2.

Chemical Information：

Molecular Weight (MW)		461.49
Formula		C23H24FN9O
CAS No.		1001350-96-4
Solubility (25°C) *	DMSO	92 mg/mL (199.35 mM)
	Water	Insoluble
	Alcohol	92 mg/mL (199.35 mM)

Biological Activity：

Targets IC50

VEGFR2 1 nM

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	2.1669 mL	10.8345 mL	21.6689 mL
5 mM	0.4334 mL	2.1669 mL	4.3338 mL
10 mM	0.2167 mL	1.0834 mL	2.1669 mL
50 mM	0.0433 mL	0.2167 mL	0.4334 mL

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