Description：

AZ6102 is a potent TNKS1/2 inhibitor that has 100-fold selectivity against other PARP family enzymes and shows IC50 of 5 nM for Wnt pathway inhibition in DLD-1 cells.

Chemical Information：

Molecular Weight (MW)		428.53
Formula		C25H28N6O
CAS No.		1645286-75-4
Solubility (25°C) *	DMSO	85 mg/mL (198.35 mM)
	Water	Insoluble
	Alcohol	Insoluble

Biological Activity：

Targets IC50

Aurora A JNK3 TRKA Flt3 JNK2 JNK1 60 nM 90 nM 70 nM 90 nM 40 nM 40 nM

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	2.3336 mL	11.6678 mL	23.3356 mL
5 mM	0.4667 mL	2.3336 mL	4.6671 mL
10 mM	0.2334 mL	1.1668 mL	2.3336 mL
50 mM	0.0467 mL	0.2334 mL	0.4667 mL

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