Description：

AS-604850 is a selective, ATP-competitive PI3Kγ inhibitor with IC50 of 250 nM, over 80-fold selectivity for PI3Kγ than PI3Kδ/β, and 18-fold more selective for PI3Kγ than PI3Kα.

Chemical Information：

Molecular Weight (MW)		285.22
Formula		C11H5F2NO4S
CAS No.		648449-76-7
Solubility (25°C) *	DMSO	57 mg/mL (199.84 mM)
	Water	Insoluble
	Alcohol	5 mg/mL (17.53 mM)

Biological Activity：

Targets IC50

B-RafV600E C-Raf SRMS FGR ACK1 MAP4K5 (KHS1) 31 nM 48 nM 18 nM 63 nM 19 nM 51 nM

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	3.5061 mL	17.5303 mL	35.0607 mL
5 mM	0.7012 mL	3.5061 mL	7.0121 mL
10 mM	0.3506 mL	1.7530 mL	3.5061 mL
50 mM	0.0701 mL	0.3506 mL	0.7012 mL

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