Description：

AS-252424 is a novel, potent PI3Kγ inhibitor with IC50 of 30 nM in a cell-free assay with 30-fold selectivity for PI3Kγ than PI3Kα, and low inhibitory activity towards PI3Kδ/β.

Chemical Information：

Molecular Weight (MW)		305.28
Formula		C14H8FNO4S
CAS No.		900515-16-4
Solubility (25°C) *	DMSO	61 mg/mL (199.81 mM)
	Water	Insoluble
	Alcohol	Insoluble

Biological Activity：

Targets IC50

mTOR PI3Kα PI3Kγ 5 nM 1.89 μM 7.37 μM

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	3.2757 mL	16.3784 mL	32.7568 mL
5 mM	0.6551 mL	3.2757 mL	6.5514 mL
10 mM	0.3276 mL	1.6378 mL	3.2757 mL
50 mM	0.0655 mL	0.3276 mL	0.6551 mL

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