Description：

Orantinib (TSU-68, SU6668) has greatest potency against PDGFR autophosphorylation with K_i of 8 nM in a cell-free assay, but also strongly inhibits Flk-1 and FGFR1 trans-phosphorylation, little activity against IGF-1R, Met, Src, Lck, Zap70, Abl and CDK2; does not inhibit EGFR. Phase 3.

Chemical Information：

Molecular Weight (MW)		310.35
Formula		C18H18N2O3
CAS No.		252916-29-3
Solubility (25°C) *	DMSO	62 mg/mL (199.77 mM)
	Water	Insoluble
	Alcohol	Insoluble

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	3.2222 mL	16.1108 mL	32.2217 mL
5 mM	0.6444 mL	3.2222 mL	6.4443 mL
10 mM	0.3222 mL	1.6111 mL	3.2222 mL
50 mM	0.0644 mL	0.3222 mL	0.6444 mL

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