Description：

Omarigliptin (MK-3102) is a competitive, reversible inhibitor of DPP-4 (IC50 = 1.6 nM, Ki = 0.8 nM). It is highly selective over all proteases tested (IC50 > 67 μM), including QPP, FAP, PEP, DPP8, and DPP9 and has weak ion channel activity (IC50 > 30 μM at IKr, Caγ1.2, and Naγ1.5).

Chemical Information：

Molecular Weight (MW)		398.43
Formula		C17H20F2N4O3S
CAS No.		1226781-44-7
Solubility (25°C) *	DMSO	79 mg/mL (198.27 mM)
	Water	Insoluble
	Alcohol	Insoluble

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	2.5099 mL	12.5493 mL	25.0985 mL
5 mM	0.5020 mL	2.5099 mL	5.0197 mL
10 mM	0.2510 mL	1.2549 mL	2.5099 mL
50 mM	0.0502 mL	0.2510 mL	0.5020 mL

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