Description：

Idelalisib (CAL-101, GS-1101) is a selective p110δ inhibitor with IC50 of 2.5 nM in cell-free assays; shown to have 40- to 300-fold greater selectivity for p110δ than p110α/β/γ, and 400- to 4000-fold more selectivity to p110δ than C2β, hVPS34, DNA-PK and mTOR.

Chemical Information：

Molecular Weight (MW)		415.42
Formula		C22H18FN7O
CAS No.		870281-82-6
Solubility (25°C) *	DMSO	83 mg/mL warmed (199.79 mM)
	Water	Insoluble
	Alcohol	23 mg/mL (55.36 mM)

Biological Activity：

Targets IC50

S1P 0.5 μM

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	2.4072 mL	12.0360 mL	24.0720 mL
5 mM	0.4814 mL	2.4072 mL	4.8144 mL
10 mM	0.2407 mL	1.2036 mL	2.4072 mL
50 mM	0.0481 mL	0.2407 mL	0.4814 mL

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