Description：

H 89 2HCl is a potent PKA inhibitor with K_i of 48 nM in a cell-free assay, 10-fold selective for PKA than PKG,500-fold greater selectivity than PKC, MLCK, calmodulin kinase II and casein kinase I/II.

Chemical Information：

Molecular Weight (MW)		519.28
Formula		C20H20BrN3O2S.2HCl
CAS No.		130964-39-5
Solubility (25°C) *	DMSO	104 mg/mL (200.27 mM)
	Water	6 mg/mL (11.55 mM)
	Alcohol	Insoluble

Biological Activity：

Targets IC50

20S proteasome β 20S proteasome 36 nM 82 nM

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	1.9257 mL	9.6287 mL	19.2574 mL
5 mM	0.3851 mL	1.9257 mL	3.8515 mL
10 mM	0.1926 mL	0.9629 mL	1.9257 mL
50 mM	0.0385 mL	0.1926 mL	0.3851 mL

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