Description：

GW4064 is an agonist of farnesoid X receptor (FXR) with EC50 of 65 nM in CV1 cell line and displays no activity at other nuclear receptors at concentrations up to 1 μM.

Chemical Information：

Molecular Weight (MW)		542.84
Formula		C28H22Cl3NO4
CAS No.		278779-30-9
Solubility (25°C) *	DMSO	100 mg/mL (184.21 mM)
	Water	Insoluble
	Alcohol	Insoluble

Biological Activity：

Targets IC50

PI3Kδ PI3Kα mTOR PI3Kα-H1047 PI3Kβ PI3Kγ 2.7 nM 2.6 nM 3.4 nM 3.3 nM 21 nM 3.0 nM

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	1.8422 mL	9.2108 mL	18.4216 mL
5 mM	0.3684 mL	1.8422 mL	3.6843 mL
10 mM	0.1842 mL	0.9211 mL	1.8422 mL
50 mM	0.0368 mL	0.1842 mL	0.3684 mL

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