Description：

GSK2606414 is an orally available, potent, and selective PERK inhibitor with IC50 of 0.4 nM, displaying at least 100-fold selectivity over the other EIF2AKs assayed.

Chemical Information：

Molecular Weight (MW)		451.44
Formula		C24H20F3N5O
CAS No.		1337531-36-8
Solubility (25°C) *	DMSO	90 mg/mL (199.36 mM)
	Water	Insoluble
	Alcohol	19 mg/mL (42.08 mM)

Biological Activity：

Targets IC50

IKK-2 3-12 μM

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	2.2151 mL	11.0757 mL	22.1513 mL
5 mM	0.4430 mL	2.2151 mL	4.4303 mL
10 mM	0.2215 mL	1.1076 mL	2.2151 mL
50 mM	0.0443 mL	0.2215 mL	0.4430 mL

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