Description：

AM251 block the inhibitory effects of endocannabinoids and synthetic cannabinoid agonists on transmitter release through an action at presynaptic cannabinoid 1 receptors in brain.

Chemical Information：

Molecular Weight (MW)		555.24
Formula		C22H21Cl2IN4O
CAS No.		183232-66-8
Solubility (25°C) *	DMSO	40 mg/mL (72.04 mM)
	Water	Insoluble
	Alcohol	Insoluble

Biological Activity：

Targets IC50

Opioid receptor δ-opioid recept κ-opioid recept 32 nM (Ki) 0.8 nM (Ki) 37  nM (Ki)

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	1.8010 mL	9.0051 mL	18.0102 mL
5 mM	0.3602 mL	1.8010 mL	3.6020 mL
10 mM	0.1801 mL	0.9005 mL	1.8010 mL
50 mM	0.0360 mL	0.1801 mL	0.3602 mL

Bought notes(bought amounts latest0)

No one bought this product

Total 0 records, divided into1 pages. First Prev Next Last