Search
Search Type: Product Name, Cat No., CAS No., Chemical Name
|
Description:
1-Azakenpaullone is a potent and selective GSK-3β inhibitor with IC50 of 18 nM, >100-fold selectivity over CDK1/cyclin B and CDK5/p25.
Chemical Information:
Molecular Weight (MW) 328.16 Formula
C15 H10 Br N3 O
CAS No. 676596-65-9 Solubility (25°C) * DMSO 66 mg/mL (201.12 mM) Water Insoluble Alcohol Insoluble
Biological Activity:
Targets IC50
Bcl-xL Bcl-2 Bcl-w ≤ 0.5 nM (Ki) ≤1 nM (Ki) ≤ 1 nM (Ki)
Preparing Stock Solutions
Concentration Volume (DMSO) Mass 1 mg 5 mg 10 mg 1 mM 3.0473 mL 15.2365 mL 30.4729 mL 5 mM 0.6095 mL 3.0473 mL 6.0946 mL 10 mM 0.3047 mL 1.5236 mL 3.0473 mL 50 mM 0.0609 mL 0.3047 mL 0.6095 mL
Bought notes(bought amounts latest0)
No one bought this product